K252A - Amerigo Scientific

- Overview
  - K252A is a staurosporine analogue isolated from a Nocardiopsis strain as a potent inhibitor of protein kinase C. K252A exhibits potent antitumor activity but shows no antimicrobial activity in vitro, or in vivo toxicity in rodents. While K252A is a potent inhibitor of Ca2+/calmodulin kinase II, it is also active against other kinases, notably myosin light chain kinase, cAMP-dependent protein kinase (PKA), protein kinase C (PKC) and cGMP-dependent protein kinase (PKG).
    
    K252A is soluble in ethanol, methanol, DMF or DMSO. Limited water solubility.
    
    Please contact us at for specific academic pricing.
- Properties
  - CAS Number
    
    99570-78-2
    
    Molecular Formula
    
    C26H19N3O5
    
    Molecular Weight
    
    453.5
    
    Appearance
    
    White solid
    
    Storage
    
    -20°C
    
    * For research use only