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Overview
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N,N'-(Sulfonyldi-4,1-phenylene)bis(2-chloroacetamide)
Selectiveprotein arginine methyltransferase 1 (PRMT1) inhibitor, IC50 = 1.5 µM. Displays no activity against CARM1 and Set7/9 methyltransferases. Inhibits growth of MCF7a breast cancer cells and LNCaP prostate cancer cells. Blocks androgen-induced gene expression in LNCaP cells.Please contact us at for specific academic pricing.
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Overview