Name: UFP 101
Price: 348.00 USD

- Overview
  - Potent and selective nociceptin receptor antagonist.
    UFP 101 is a potent, selective and competitive antagonist at the nociceptin receptor. UFP 101 binds to nociceptin receptors with high affinity (pKi 10.24) and possesses ~3000 fold selectivity over the classical opioid receptors. UFP 101 is antinociceptive and opposes the action of nociceptin in vivo, with an antinociceptive effect when given i.c.v. while being inactive following spinal administration in mice. UFP 101 also shows antidepressant effects in distinct species and can reduce microvascular inflammation to lipopolysaccharide in vivo.
    
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- Properties
  - Categories
    
    Peptides
    
    Alternative Name
    
    [Nphe1,Arg14,Lys15]nociceptin-NH2, [Nphe1, Arg14, Lys15] N/OFQ NH2
    
    Molecular Formula
    
    C82H138N32O21
    
    Molecular Weight
    
    1908.19
    
    Appearance
    
    Freeze dried solid
    
    Purity
    
    >95% by HPLC
    
    Solubility
    
    Soluble to 1 mg/ml in water
    
    Other Properties
    
    Sequence: Bn-Gly-Gly-Gly-Phe-Thr-Gly-Ala-Arg-Lys-Ser-Ala-Arg-Lys-Arg-Lys-Asn-Gln-NH2,Bn-GGGFTGARKSARKRKNQ-NH2
    Modification: N-terminal benzyl, C-terminal amide
    
    Storage
    
    Store dry, frozen and in the dark
    
    * Please note: this product can only be supplied to registered research and development facilities, and may be used for in vitro research use only, not for administration to humans or animals.

UFP 101

UFP 101

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