Name: Varenicline Tartrate
Price: 212.00 USD

- Overview
  - Please contact us at for specific academic pricing.
    
    Background
    
    Orally active, subtype-selective partial agonist at α4β2 nicotinic receptors (Ki values are 0.06, 240, 322 and 3540 nM for α4β2, α3β4, α7, α1βγδ receptors respectively). Reduces nicotine-evoked dopamine release in vitro and decreases nicotine self-adminis
- Properties
  - Categories
    
    Subtype-selective agonist of α4β2 nicotinic receptors, orally active
    
    Alternative Name
    
    (6R)-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline (2R,3R)-2,3-dihydroxysuccinate
    
    CAS Number
    
    375815-87-5
    
    Molecular Formula
    
    C13H13N3·C4H6O6
    
    Molecular Weight
    
    361.35
    
    Appearance
    
    A solid
    
    Purity
    
    98.52%
    
    Solubility
    
    insoluble in EtOH; ≥18.07 mg/mL in DMSO; ≥96.2 mg/mL in H2O
    
    Storage
    
    Store at -20°C
    
    SMILES
    
    O=C([[email protected]]([[email protected]@](C(O[H])=O)([H])O[H])([H])O[H])O[H].[H][[email protected]@]12C([H])([H])C(C([H])([H])N([H])C2([H])[H])([H])C3=C([H])C4=NC([H])=C([H])N=C4C([H])=C13
    
    * For Research Use Only