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Alvimopan

Alvimopan

Catalog Number:

L002368510APE

Mfr. No.:

APE-A3162

Price:

$252

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- Overview
  - Please contact us at for specific academic pricing.
    
    Background
    
    Alvimopan(ADL 8-2698; Entereg; LY 246736) is a selective and competitive antagonist at mu-opioid receptors, found in myenteric and submucosal neurons and the immune cells of the lamina propria in the human gut. Upon administration, Alvimopan(ADL 8-2698; Entereg; LY 246736) binds to mu-opioid receptors in the gut, thereby reversing opiod-related disturbances in gut motility. Alvimopan is approximately three to nine times more potent than naloxone.A synthetic trans-3,4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity.
- Properties
  - Categories
    
    Mu-opioid receptors antagonist
    
    Alternative Name
    
    ADL 8-2698; Entereg; LY 246736; 2-((Z)-((S)-2-benzyl-1-hydroxy-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propylidene)amino)acetic acid
    
    CAS Number
    
    156053-89-3
    
    Molecular Formula
    
    C25H32N2O4
    
    Molecular Weight
    
    424.53
    
    Purity
    
    98.00%
    
    Solubility
    
    insoluble in H2O; insoluble in EtOH; ≥25.7 mg/mL in DMSO
    
    Storage
    
    Store at -20°C
    
    SMILES
    
    C[[email protected]@]1([H])CN(C[[email protected]](/C(O)=N/CC(O)=O)([H])CC2=CC=CC=C2)CC[[email protected]]1(C3=CC(O)=CC=C3)C
    
    * For Research Use Only

Documents

COA (Certificate Of Analysis)

MSDS (Material Safety Data Sheet)

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