1,3,4,5-Tetramethyl-2-[(2-oxopropyl)thio]imidazolium chloride

- Overview
  - T101 (L-682.777) is a good blocker of tissue transglutaminase and coagulation factor XIIIa. Both enzymes are inhibited with an IC50 of about 0.25 μM.
    
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    More Details
    
    Zedira
- Properties
  - Molecular Weight
    
    248,77
    
    Storage
    
    Store at -20°C
    
    * Intended for research use only, not for use in human, therapeutic or diagnostic applications.
- Applications
  - Application
    
    FXIII Inhibitors
    
    Application Description
    
    Inhibitor for transglutaminase.The molecule was developed to block coagulation factor XIIIa, however the compound inhibits tissue transglutaminase as well. Both enzymes are inhibited with an IC50 of about 0.25 μM.
- Reference
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