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Terfenadine

Terfenadine

Catalog Number:
L002369600APE
Mfr. No.:
APE-A8534
Price:
$196
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      • Overview

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          Background

          Terfenadine is a histamine H1-receptor antagonist, which blocks HERG and KATP (KIR6) channels. The IC values for Terfenadines inhibitory activity against these channels is 204nM for HERG and 1.2µM for KATP. Studies show that Terfenadine inhibits the delayed rectifier K+ in ventricular myocytes. Terfenadine is converted into its more active form, terfenadine carboxylate by the enzyme CYP3A4.

      • Properties
        • Categories
          Histamine H1-receptor antagonist
          Alternative Name
          1-(4-tert-butylphenyl)-4-[4-[hydroxy(diphenyl)methyl]piperidin-1-yl]butan-1-ol
          CAS Number
          50679-08-8
          Molecular Formula
          C32H41NO2
          Molecular Weight
          471.67
          Appearance
          A solid
          Purity
          98.00%
          Solubility
          insoluble in H2O; ≥18 mg/mL in DMSO; ≥8.06 mg/mL in EtOH with ultrasonic
          Storage
          Store at -20°C
          SMILES
          CC(C)(C)C1=CC=C(C=C1)C(CCCN2CCC(CC2)C(C3=CC=CC=C3)(C4=CC=CC=C4)O)O

          * For Research Use Only

    Documents

    COA (Certificate Of Analysis)

    MSDS (Material Safety Data Sheet)

    Datasheet

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